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| Product Name | AKR1C1 Inhibitor, 5-PBSA |
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| Description | Purity ~94% (HPLC). A cell-permeable salicylic acid compound that acts as a highly potent, active-site directed and substrate competitive AKR1C1 inhibitor (Ki=4nM) with moderate to excellent selectivity over AKR1C2, AKR1C3 and AKR1C4 (Ki=0.087, 4.2 and 18.2uM, respectively). Shown to inhibit the metabolism of progesterone by AKR1C1 (IC50=460nM in AKR1C1 overexpressing BAECs). Solubility: DMSO NMR: Conforms LC-MS: Conforms |
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| Size | 25mg |
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| Concentration | n/a |
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| Applications | n/a |
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| Other Names | AKR1C1 Inhibitor, 5-PBSA (Aldo-Keto Reductase Family 1 Member C1 Inhibitor, 5-PBSA, 3-Bromo-5-phenylsalicylic Acid, 20a-Hydroxysteroid Dehydrogenase Inhibitor, 5-PBSA) |
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| Gene, Accession, CAS # | n/a |
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| Catalog # | 217167 |
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| Order / More Info | AKR1C1 Inhibitor, 5-PBSA from UNITED STATES BIOLOGICAL |
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| Product Specific References | n/a |
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