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| Product Name | Flumazenil (GABAA Receptor Antagonist, Flumazenil, Ro 15-1788) |
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| Description | Purity ~99% (HPLC). A competitive blocker of benzodiazepine activation of inhibitory GABAergic synpases (ID50 = 200ug/kg/i.p). Binds to the benzodiazepine site of GABAA receptors. Enhances GABAA-receptor mediated currents and antagonizes the enhancing effects of benzodiapine agonist flurazepam. Exhibits fast association and dissociation from the benzodiazepine binding site. Permeates the blood brain barrier, however, the level of uptake may depend on efflux effects of p-glycogprotein transporter. Solubility: DMSO Primary Target: GABA-A |
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| Size | 10mg |
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| Concentration | n/a |
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| Applications | n/a |
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| Other Names | n/a |
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| Gene, Accession, CAS # | n/a |
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| Catalog # | 217359 |
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| Order / More Info | Flumazenil (GABAA Receptor Antagonist, Flumazenil, Ro 15-1788) from UNITED STATES BIOLOGICAL |
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| Product Specific References | n/a |
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