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| Product Name | G-1 |
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| Description | G-1 is a potent and selective G protein-coupled estrogen receptor (GPER) agonist (Ki = 11 nM, EC50 = 2 nM); displays no activity at ERα and ERβ at concentrations up to 10 µM. Increases cytosolic Ca2+ and inhibits migration of SKBr3 cells and MCF-7 cells in response to chemoattractants (IC50 values are 0.7 and 1.6 nM respectively) in vitro. Blocks MCF-1 cell cycle progression at the G1 phase. Displays therapeutic effects in the mouse EAE model of multiple sclerosis. Molecular Formula: C21H18BrNO3 Solubility: DMSO (Slightly), Methanol (Slightly, Heated) Molecular Weight: 412.28 |
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| Size | 1mg, 2.5mg |
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| Concentration | n/a |
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| Applications | n/a |
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| Other Names | n/a |
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| Gene, Accession, CAS # | n/a |
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| Catalog # | 451022 |
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| Order / More Info | G-1 from UNITED STATES BIOLOGICAL |
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| Product Specific References | n/a |
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