| 产品详情 |
| Edit |   |
|---|
| Product Name | Adenosine A2B Receptor Antagonist I, MRS 1754 |
|---|
| Description | Purity ~99% (HPLC). A p-cyanoanilide xanthine derivative that acts as a highly selective, high affinity antagonist of adenosine A2B receptor (A2BR; Ki = 1.97nM for human A2BR). Does not significantly affect other adenosine receptors (Ki = 403nM, 503nM, and 570nM for human A1R, A2AR, and A3R, respectively). Exhibits some antagonist action on rat A1R (Ki = 16.8nM). Shown to abolish the cardioprotective effects of NECA. Primary Target: Adenosine A2B Receptor Primary Target Ki: 1.97nM Molar Mass: 486.5 Solubility: DMSO |
|---|
| Size | 10mg |
|---|
| Concentration | n/a |
|---|
| Applications | n/a |
|---|
| Other Names | Adenosine A2B Receptor Antagonist I, MRS 1754 (8-[4-[((4-Cyanophenyl)carbamoylmethyl)oxy]phenyl]-1,3-di(n-propyl)xanthine, MRS-1754, MRS1754) |
|---|
| Gene, Accession, CAS # | n/a |
|---|
| Catalog # | 217155 |
|---|
| Price | |
|---|
| Order / More Info | Adenosine A2B Receptor Antagonist I, MRS 1754 from UNITED STATES BIOLOGICAL |
|---|
| Product Specific References | n/a |
|---|
| 产品资料 |
|
|